Sunday, October 16, 2016

Lubiprostone Pharmacokinetics


Unlike abounding laxative products, lubiprostone does not appearance signs of tolerance, dependency, or adapted serum electrolyte concentration. There was no backlash aftereffect afterward abandonment of treatment, but a bit-by-bit acknowledgment to pre-treatment bowel movement abundance should be expected.
Minimal administration of the biologic occurs above the actual gastrointestinal tissues. Lubiprostone is rapidly metabolized by reduction/oxidation, advised by carbonyl reductase. There is no metabolic captivation of the hepatic cytochrome P450 system. The assessable metabolite, M3, exists in actual low levels in claret and makes up beneath than 10% of the absolute administered dose.

Data announce that metabolism occurs locally in the abdomen and jejunum.

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